
CaM kinase II inhibitor TFA salt
CAS No. ——
CaM kinase II inhibitor TFA salt( Autocamtide-2-related inhibitory peptide (TFA) )
Catalog No. M22306 CAS No. ——
Autocamtide-2-Related Inhibitory Peptide is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.It is found that Autocamtide-2-related inhibitory peptide (TFA) is a potent inhibitor of CaM-kinase II with an IC50 of 40 nM, which is active in the presence or absence of Ca2+/calmodulin.
Purity : >98% (HPLC)






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Biological Information
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Product NameCaM kinase II inhibitor TFA salt
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NoteResearch use only, not for human use.
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Brief DescriptionAutocamtide-2-Related Inhibitory Peptide is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.It is found that Autocamtide-2-related inhibitory peptide (TFA) is a potent inhibitor of CaM-kinase II with an IC50 of 40 nM, which is active in the presence or absence of Ca2+/calmodulin.
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DescriptionAutocamtide-2-Related Inhibitory Peptide is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.It is found that Autocamtide-2-related inhibitory peptide (TFA) is a potent inhibitor of CaM-kinase II with an IC50 of 40 nM, which is active in the presence or absence of Ca2+/calmodulin. It is 50 and 500 times more potent than CaMK-(281-302Ala286) and KN-93, respectively, under the assay condition used.
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In Vitro——
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In Vivo——
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SynonymsAutocamtide-2-related inhibitory peptide (TFA)
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PathwayEndocrinology/Hormones
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TargetCaMK
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RecptorCaMKII
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Research Area——
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Indication——
Chemical Information
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CAS Number——
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Formula Weight1611.76
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Molecular FormulaC66H126N22O21F3
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Purity>98% (HPLC)
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Solubility——
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SMILESC[C@H](NC(=O)[C@@H](NC(=O)[C@@H](N)CCCCN)CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@@H](C)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC(C)C)C(O)=O.FC(F)(F)C(=O)O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Ishida A, et al. A novel highly specific and potent inhibitor of calmodulin-dependent protein kinase II. Biochem Biophys Res Commun. 1995 Jul 26;212(3):806-12.
molnova catalog



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